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I-β-Nicotinamide Adenine Dinucleotide Phosphate Disodium Salt CAS:24292-60-2
β-Nicotinamide Adenine Dinucleotide Phosphate Disodium Saltiyi-coenzyme esakazeka kabanzi ezintweni eziphilayo, Ihlanganyela ekwehliseni i-oxidation. Isebenza njengomthwali we-electron ekwelashweni okuningana, i-oxidized alternately (NADP+) kanye ne-decresed (NADPH).β-Nicotinamide Adenine Dinucleotide Phosphate Disodium Saltiyinto lapho i-nicotinic acid amide adenine dinucleotide kanye ne-molecule ye-phosphate ziboshwe khona yi-ester bond. Iyi-hydrogen receptor futhi ingasetshenziswa ekuthuthukiseni nasekuthuthukiseni izinhlobo ezahlukene ze-reagents zokuxilonga ze-in vitro.
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I-β-Nicotinamide Adenine Dinucleotide Lithium usawoti (NAD Lithium salt) CAS:64417-72-7
β-Nicotinamide Adenine Dinucleotide Usawoti we-lithiumiyi-coenzyme ebalulekile ekusebenzeni kwe-metabolism. Etholakala kuwo wonke amaseli aphilayo, i-NAD ibizwa ngokuthi i-dinucleotide ngoba iqukethe ama-nucleotide amabili ahlanganiswe ngamaqembu awo e-phosphate. I-nucleotide eyodwa iqukethe i-adenine nucleobase kanti enye i-nicotinamide. I-NAD ikhona ngezindlela ezimbili: ifomu elihlanganisiwe nelincishisiwe, elifushanisiwe njenge-NAD+ kanye ne-NADH (H ye-hydrogen), ngokulandelana.
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I-Venlafaxine CAS:93413-69-5
I-Venlafaxine iyisidakamizwa sokucindezeleka sesigaba se-serotonin kanye ne-norepinephrine reuptake inhibitor (SNRI). Lesi sidakamizwa saqala ukwenziwa nguWyeth ku-19Chemicalbook93 futhi manje sithengiswa yi-Pfizer. Lesi sidakamizwa sivunyelwe ukwelapha isifo sokucindezeleka esikhulu (MDD), isifo sokukhathazeka esijwayelekile (GAD), kanye nokucindezeleka okuhambisana nokukhathazeka.
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Umhlinzeki Womkhiqizi we-Ciclopirox Ethanolamine CAS:41621-49-2
I-Ciclopirox ethanolamine iyi-ejenti yokulwa ne-gfungal ene-spectrum ebanzi, futhi ikhombisa umsebenzi wokulwa namagciwane ngokumelene namagciwane amaningi e-Gram-positive kanye ne-Gram-negative, futhi inezakhiwo zokulwa nokuvuvukala. Isetshenziswa njengokwelashwa kwesikhumba se-fungus kanye nokutheleleka kwezinzipho.
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I-Desvenlafaxine Succinate CAS:386750-22-7
I-Desvenlafaxine Succinate iyi-dual serotonin kanye ne-norepinephrine reuptake inhibitor (SNRI) eyavunyelwa ukwelapha isifo sokucindezeleka okukhulu (MDD) e-United States ngo-2008. Ukuze kuthuthukiswe ukusebenza kahle kanye nephrofayili yokuphepha ye-venlafaxine, uWyeth wathola futhi wakha enye yama-metabolite amakhulu e-venlafaxine, okuyi-O-desmethyl metabolite (desvenlafaxine).
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I-Doxazosin Mesylate CAS: 77883-43-3 Umhlinzeki Womkhiqizi
I-Doxazosin mesylate iyinhlanganisela ye-quinazoline eyisivimbeli esikhethiwe se-alpha1 subtype yama-alpha adrenergic receptors. I-Doxazosin mesylate iyisizukulwane esisha se-quinazolone α1 receptor blocker esakhiwe yinkampani i-Pfizer (e-United States). Inesikhathi eside sokuphila, isebenzisa imiphumela yayo yokwandisa imithambo yegazi, ukunciphisa ukumelana kwemithambo yegazi kanye nokwehlisa umfutho wegazi ngokuvimbela i-a1 receptor. Inconywe kwamanye amazwe njengemithi yokuqala yokwelapha yomugqa wokulwa nomfutho wegazi ophakeme kanye nokwelashwa kwesifo se-prostate.
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Umhlinzeki Womkhiqizi we-L-Isoleucine CAS: 73-32-5
I-L-Isoleucine, eyaziwa nangokuthi i-Isoleucine, iyi-amino acid eyi-isomer ye-leucine. Ibalulekile ekwakhiweni kwe-hemoglobin kanye nokulawulwa kwamazinga kashukela kanye namandla egazini. I-L-Isoleucine iyi-isomer ye-L-leucine futhi iyi-amino acid ebalulekile. Yenziwe kusuka ku-threonine futhi iyi-amino acid eyi-branched-chain hydrophobic.
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I-Captopril CAS: 62571-86-2 Umhlinzeki Womkhiqizi
I-Captopril iyisidakamizwa esifundwa kakhulu phakathi kwezidakamizwa eziguqula i-angiotensin eziphakanyiswa njengomuthi wokunciphisa umfutho wegazi. Ivimba i-enzyme eguqula i-angiotensin, evimbela ukwakheka kwe-angiotensin II futhi inciphise umphumela wayo wokunciphisa imithambo yegazi emikhunjini yemithambo yegazi neyemithambo yegazi. Ukucindezeleka kwemithambo yegazi yonke kuyancipha, okuholela ekwehleni komfutho wegazi.
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Umhlinzeki Womkhiqizi weCandesartan CAS:139481-59-7
I-Candesartan iyi-angiotensin II receptor I (AT1) antagonist, i-IC50s=1.12 kanye ne-2.86 nM ye-bovine adrenal cortex kanye ne-rabbit aorta ngokulandelana. Ivimbela ngokukhetha ukufinyela okubangelwa yi-angiotensin II kwemigqa ye-rabbit aortic ngaphandle kokuthinta ukufinyela okubangelwa ezinye izinto ezifana ne-norepinephrine, i-KCl, i-serotonin, i-PGF2α noma i-endothelin.
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I-Candesartana Cilexetila CAS:145040-37-5
I-Candesartan Celexetil iyi-ester analog ye-angiotensin II antagonist i-Candesartan (sc-217825). Ukuphikisana kwale receptor kuvimbela ukubopha kwe-angiotensin II, i-vasoconstrictor enamandla. Lokhu kunomphumela ojwayelekile wokwanda kwe-vasodilation kanye nomthamo wegazi okhuphukile. I-Candesartan Celexetil Ester iyisithibi se-AT1.
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Umhlinzeki Womkhiqizi we-Bupropion CAS: 34911-55-2
I-Bupropion iyi-aromatic ketone eyi-propiophenone ephethe iqembu le-tert-butylamino endaweni yesi-2 kanye ne-chloro substituent endaweni yesi-3 eringini ye-phenyl. Inendima njengomphilisi wokudambisa ukucindezeleka, ukungcola kwemvelo kanye ne-xenobiotic. Iyi-amino compound yesibili, ilungu le-monochlorobenzenes kanye ne-aromatic ketone.
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I-Bezafibrate CAS:41859-67-0 Umhlinzeki Womkhiqizi
I-Bezafibrate iyi-monocarboxylic acid amide etholakala ngokujiya okusemthethweni kweqembu le-carboxy le-4-chlorobenzoic acid neqembu lama-amino le-2-[4-(2-aminoethyl)phenoxy]-2-methylpropanoic acid. I-Benafibrate isetshenziselwa ukwelapha i-hyperlipidaemia. Inendima njenge-xenobiotic, i-contaminant yemvelo, i-geroprotector kanye nomuthi we-antilipemic. Iyi-monocarboxylic acid, i-aromatic ether, ilungu le-monochlorobenzenes kanye ne-monocarboxylic acid amide. Ihlobene ngokusebenza ne-propionic acid.
