Ibhande Nomgwaqo: Ukubambisana, Ukuzwana kanye Nokunqoba Nokunqoba
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Amakhemikhali Ahle

  • 5-Bromo-2-chloro-4-(cyclopentylamino)pyrimidine CAS:733039-20-8

    5-Bromo-2-chloro-4-(cyclopentylamino)pyrimidine CAS:733039-20-8

    5-I-Bromo-2-chloro-4-(cyclopentylamino)pyrimidine iyinhlanganisela yamakhemikhali ecwaningwa ocwaningweni lwezemithi. Inesakhiwo se-pyrimidine esinokushintshwa kwe-bromo ne-chloro, okungenzeka kube usizo ekusetshenzisweni kwezokwelapha, kugxilwe ezindleleni ezithile zesifo noma ezindleleni zebhayoloji ekutholakaleni kwemithi.

     

  • 4-[6-[[6-(1-Butoxyvinyl)-8-cyclopentyl-5-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl]amino]pyridin-3-yl]piperazine-1-carboxylic acid tert-butyl ester CAS:866084-31-3

    4-[6-[[6-(1-Butoxyvinyl)-8-cyclopentyl-5-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl]amino]pyridin-3-yl]piperazine-1-carboxylic acid tert-butyl ester CAS:866084-31-3

    4-[6-[[6-(1-Butoxyvinyl)-8-cyclopentyl-5-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl]amino]pyridin-3-yl]piperazine-1-carboxylic acid i-tert-butyl ester iyinhlanganisela yamakhemikhali eyinkimbinkimbi equkethe umgogodla we-piperazine onamaqembu asebenzayo afaka phakathi i-pyridine, i-pyrimidine, kanye ne-tert-butyl ester. Isakhiwo sayo sisekela ukusetshenziswa okungenzeka kumakhemikhali ezokwelapha kanye nokuthuthukiswa kwemithi ngenxa yezinhlobo zayo ezahlukene ze-pharmacophores.

     

  • I-Bortezomib CAS:179324-69-7

    I-Bortezomib CAS:179324-69-7

    I-Bortezomib iyinhlanganisela yemithi esetshenziswa ekwelapheni i-multiple myeloma kanye ne-mantle cell lymphoma. Ingesigaba sama-proteasome inhibitors, ehlose ama-enzyme e-proteolytic emaselini ukuphazamisa ukusebenza kwawo futhi ibangele i-apoptosis (ukufa kweseli okuhleliwe). Le ndlela iyenza isebenze kahle ngokumelene nomdlavuza othile lapho ukukhula kweseli okungalawulwa kwenzeka khona.

  • I-Methyl 2-bromomethyl-3-nitrobenzoate CAS:98475-07-1

    I-Methyl 2-bromomethyl-3-nitrobenzoate CAS:98475-07-1

    I-Methyl 2-bromomethyl-3-nitrobenzoate iyinhlanganisela yamakhemikhali equkethe iqembu le-nitro endaweni engu-3 kanye neqembu le-bromomethyl endaweni engu-2 yomgogodla we-benzoate. Isetshenziswa ekwakhiweni kwezinto eziphilayo njengendlela eguquguqukayo, evumela ukwakhiwa kwama-molecule ayinkimbinkimbi anamaqembu athile asebenzayo.

  • I-Pemetrexed disodium INT-5 CAS:165049-28-5

    I-Pemetrexed disodium INT-5 CAS:165049-28-5

    I-Pemetrexed disodium INT-5 umuthi we-oncology ohlukaniswe ngaphansi kwama-antifolate chemotherapy agents. Isetshenziswa kakhulu ekwelapheni umdlavuza ohlukahlukene, okuhlanganisa i-mesothelioma, umdlavuza wamaphaphu ongewona amangqamuzana amancane, kanye nomdlavuza othize osakazeka kalula.

  • I-Pemetrexed disodium INT-4 CAS:137281-39-1

    I-Pemetrexed disodium INT-4 CAS:137281-39-1

    I-Pemetrexed disodium INT-4 iyi-antifolate chemotherapy esetshenziswa ku-oncology. Isetshenziswa ekwelapheni umdlavuza ohlukahlukene, okuhlanganisa i-mesothelioma, umdlavuza wamaphaphu ongewona amangqamuzana amancane, kanye nomdlavuza othize osakazeka kalula.

  • I-Pemetrexed disodium INT-3 CAS:155405-80-4

    I-Pemetrexed disodium INT-3 CAS:155405-80-4

    I-Pemetrexed disodium INT-3 iyi-antifolate chemotherapy esetshenziswa ku-oncology. Isetshenziswa ekwelapheni umdlavuza ohlukahlukene, okuhlanganisa i-mesothelioma, umdlavuza wamaphaphu ongewona amangqamuzana amancane, kanye nomdlavuza othize osakazeka kalula.

  • Isisekelo se-Terbinafine CAS:91161-71-6

    Isisekelo se-Terbinafine CAS:91161-71-6

    Isisekelo se-Terbinafine siyisithako esisebenzayo semithi esetshenziselwa ukwelapha izifo zesikhunta. Singesigaba se-allylamine semithi elwa namagciwane futhi saziwa ngokusebenza kwayo ngokumelene nama-dermatophyte, imvubelo, kanye nezikhunta.

  • 2-Chloro-4,6-dimethoxy-1,3,5-triazine CAS:3140-73-6

    2-Chloro-4,6-dimethoxy-1,3,5-triazine CAS:3140-73-6

    2-I-Chloro-4,6-dimethoxy-1,3,5-triazine iyinhlanganisela yamakhemikhali esetshenziswa njengesakhiwo esiguquguqukayo ezinqubweni zokwenziwa kwezinto eziphilayo kanye nokuguqulwa kwamakhemikhali. Iqukethe amaqembu asebenzayo e-chloro kanye ne-methoxy anamathele esakhiweni sendandatho ye-triazine, okwenza kube lula ukusetshenziswa kwayo ekusabeleni kwamakhemikhali okuhlukahlukene kanye nokwakheka kwamakhemikhali.

     

  • I-2-Amino-4,5-bis(2-methoxyethoxy)benzonitrile CAS:950596-58-4

    I-2-Amino-4,5-bis(2-methoxyethoxy)benzonitrile CAS:950596-58-4

    2-I-Amino-4,5-bis (2-methoxyethoxy)benzonitrile iyinhlanganisela yamakhemikhali esetshenziswa ocwaningweni lwezemithi, ebonakala ngesakhiwo se-benzonitrile esine-amino kanye ne-methoxyethoxy substitutions, okungenzeka ukuthi ibalulekile ekusetshenzisweni okuthile kokwelapha.

  • (1R)-(S)-pinanediol-1-Ammonium Trifluoroacetate-3-methlbutane-1-boronate CAS:179324-87-9

    (1R)-(S)-pinanediol-1-Ammonium Trifluoroacetate-3-methlbutane-1-boronate CAS:179324-87-9

    (1R)-(S)-Pinanediol-1-Ammonium Trifluoroacetate-3-Methylbutane-1-Boronate iyinhlanganisela yamakhemikhali ebonakala ngesakhiwo esiyinkimbinkimbi esinomgogodla we-pinanediol, iqembu le-ammonium trifluoroacetate, kanye nokusebenza kwe-boronate ester. Isetshenziswa ekwakhiweni kwezinto eziphilayo njengebhloko yokwakha i-chiral, okuvumela ukudalwa kwamakhemikhali athile kanye nezidakamizwa ezisetshenziswa emithini.

  • I-Diethyl L-glutamate hydrochloride CAS:1118-89-4

    I-Diethyl L-glutamate hydrochloride CAS:1118-89-4

    I-Diethyl L-glutamate hydrochloride iyinhlanganisela yamakhemikhali esetshenziswa ngokuyinhloko njenge-synthetic intermediate ocwaningweni lwezemithi kanye nokwakheka kwezinto eziphilayo. Itholakala ku-L-glutamic acid futhi isebenza njengesandulela ekukhiqizweni kwemithi ehlukahlukene kanye namakhemikhali asebenzayo ngokwezinto eziphilayo.