Ibhande Nomgwaqo: Ukubambisana, Ukuzwana kanye Nokunqoba Nokunqoba
imikhiqizo

Imikhiqizo

I-Olmesartan CAS:144689-24-7 Umhlinzeki Womkhiqizi

I-Olmesartan medoxomil,phenyl]phenyl]methyl]imidazole-4-carboxylate (iBenicar, i-Olmetec) isebenzisa uhlelo lwe-tetrazolering njengohlelo lwayo lwe-acidic, olubamba iqhaza ekubopheni kwama-receptor. Uma inikezwa isiguli, umuthi usebenza ngokushesha nangokuphelele yi-ester hydrolysis ye-medoxomil ngesikhathi sokumuncwa kusuka emgodini wesisu. I-Olmesartan iyi-biphenylyltetrazole. Inendima njenge-ejenti yokulwa nomfutho wegazi ophakeme kanye ne-angiotensin receptor antagonist.


Imininingwane Yomkhiqizo

Amathegi Omkhiqizo

Ukusetshenziswa kanye Nomphumela

I-Omesartan iyi-antagonist ephumelelayo nekhethayo ye-AT2. I-Omesartan axetil inomphumela oqinile wokulwa nomfutho wegazi ophezulu. Ngemva kokusetshenziswa ngomlomo, ikhishwa ngokuphelele odongeni lwamathumbu amancane bese iguqulwa ibe yi-metabolite esebenzayo i-Olmesartan. I-Olmesartan iyi-antagonist ye-angiotensin II receptor engakhethi ngamakhemikhali evimbela ngokukhetha ukubopha kwe-angiotensin II kuma-receptor e-AT1 emisipha ebushelelezi yemithambo yegazi, ngaleyo ndlela ivimbele umphumela we-vasoconstrictive we-angiotensin II.

Isampula Yomkhiqizo

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Ukupakisha Umkhiqizo:

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Ulwazi Olwengeziwe:

Ukwakheka C30H32N6O6
Ukuhlolwa 99%
Ukubukeka Impuphu emhlophe
Inombolo ye-CAS 144689-24-7
Ukupakisha 25KG
Impilo Yeshelufu iminyaka engu-2
Isitoreji Gcina endaweni epholile neyomile
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