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I-Degarelix CAS:214766-78-6
I-Degarelix iyi-modulator yama-hormone esetshenziswa kakhulu ukwelapha umdlavuza we-prostate futhi yehlisa amazinga e-androgen emadodeni ngokuvimbela ukukhishwa kwama-hormone e-pituitary.
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I-Kisspeptin-10, i-CAS yomuntu: 374675-21-5
I-Kisspeptin-10, yomuntu, iyi-neuropeptide eyingxenye yomndeni wakwaKisspeptin futhi ilawula izinqubo zomzimba ezifana nokukhishwa kwama-hormone ocansi kanye nomsebenzi wokuzala ngokusebenzisa ama-receptor e-Kisspeptin.
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I-Cilengitide CAS:188968-51-6
I-Cilengitide iyisivimbeli se-integrin esivimba i-angiogenesis kanye nokusabalala kwamaseli esimila ngokuvimbela umsebenzi wama-integrin receptors.
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I-Dulaglutide CAS:923950-08-7
I-Dulaglutide iyi-peptide-1 (GLP-1) receptor agonist esetshenziswa ukwelapha isifo sikashukela sohlobo 2. Isiza ukulawula amazinga kashukela egazini ngokuvuselela ukukhishwa kwe-insulin nokunciphisa ukukhishwa kwe-glucagon, okuholela ekuthuthukisweni kokulawulwa kwe-glycemic. I-Dulaglutide inikezwa ngomjovo ongaphansi kwesikhumba kanye ngesonto futhi ivame ukunikezwa ngokuhlanganiswa nokudla kanye nokuzivocavoca ukuze kuthuthukiswe ukuphathwa kwesifo sikashukela.
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I-Bivalirudin CAS:128270-60-0
I-Bivalirudin iyi-anticoagulant evimbela ngqo umsebenzi we-thrombin egazini. Iyisivimbeli se-thromboxane esiqondile esenziwe ngendlela efana ne-thromboxane. I-Bivalirudin ayidingi i-metabolism emzimbeni ukuze ifinyelele imiphumela ye-anticoagulant futhi inemiphumela ye-anticoagulant eguqukayo.
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I-Eptifibatide CAS:188627-80-7
I-Eptifibatide umuthi ovimbela ama-platelet osetshenziselwa ukuvimbela izehlakalo zenhliziyo ezifana nokuphazamiseka kwenhliziyo kanye ne-thrombosis. Ingumphikisi we-GPIIb/IIIa receptor onciphisa i-thrombosis ngokuvimbela ukuhlangana kwama-platelet.
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I-CAS ye-Icatibant:130308-48-4
I-Icatibant umuthi we-peptide wokwenziwa oyindlela yokwelapha ekhethiwe ye-angioedema ezuzwe njengefa ebangelwa ukutheleleka yigciwane le-brucella.
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I-Ganirelix CAS:123246-29-7
I-Ganirelix iyi-peptide yokwenziwa esetshenziswa kwezokwelapha zokuzala ukuvimbela ukuvuthwa kweqanda ngaphambi kwesikhathi kwabesifazane abasebenzisa izinqubo zobuchwepheshe bokuzala ezisizayo njengokukhulelwa kwe-in vitro (IVF). Isebenza ngokuvimbela ukwanda kwe-luteinizing hormone (LH) ebangela ukuvuthwa kweqanda.
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I-Elcatonin CAS:60731-46-6
I-Elcatonin iyi-analog yokwenziwa ye-salmon calcitonin, i-peptide hormone esetshenziswa ekwelapheni izimo ezibonakala ngokumuncwa kwamathambo ngokweqile, njenge-osteoporosis nesifo sikaPaget. Isebenza ngokuvimbela umsebenzi we-osteoclast, ngaleyo ndlela inciphise ukulahleka kwamathambo futhi isize ekugcineni ubuningi bamathambo.
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I-Cetrorelix CAS:120287-85-6
I-Cetrorelix iyi-peptide yokwenziwa esetshenziswa kubuchwepheshe bokusiza ekuzaleni ukuvimbela ukuvuthwa kweqanda ngaphambi kwesikhathi ngesikhathi sokuvuselelwa kwe-ovarian okulawulwayo kwabesifazane abathatha izinqubo zokukhulelwa kwe-in vitro (IVF) ngokuvimbela ukukhishwa kwe-luteinizing hormone (LH).
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I-Carperitide CAS: 89213-87-6
I-Carperitide iwuhlobo lokwenziwa lwe-atrial natriuretic peptide (ANP), esetshenziselwa ukwelapha ukwehluleka kwenhliziyo okukhulu. Isebenza njenge-vasodilator kanye ne-diuretic ukuze ithuthukise ukusebenza kwenhliziyo futhi inciphise izimpawu ezigulini ezibhekene nokwanda okukhulu kokwehluleka kwenhliziyo.
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I-Ornipressin CAS:3397-23-7
I-Ornipressin iyisidakamizwa sokwenziwa esingeyona i-adrenergic esinemiphumela ye-vasoconstrictive futhi ifana nesakhiwo sama-hormone e-antidiuretic.
