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imikhiqizo

Imikhiqizo

I-Pitavastatin CAS:147511-69-1 Umhlinzeki Womkhiqizi

I-Pitavastatin iyisithiyo se-HMG-CoA reductase esikhuthaza isinyathelo sokuqala sokwenziwa kwe-cholesterol. Ibonakala ingenaphunga futhi imhlophe kuya ku-powder ophuzi okhanyayo. Iba nemiphumela ngokunciphisa izinga lezinto ezithile ezinamafutha njenge-cholesterol emzimbeni. Ngakho-ke, ihloselwe kakhulu ukwelapha i-hypercholesterolaemia kanye nokuvimbela izifo zenhliziyo. Ayikwazi nje ukwehlisa i-cholesterol ephezulu kanye ne-triglyceride ezigulini ezithile, kodwa futhi ingakhuphula okuqukethwe yi-high density lipoprotein (HDL), amazinga e-cholesterol "amahle". Kufanele inikezwe ngokujwayelekile kanye nokudla okufanele.


Imininingwane Yomkhiqizo

Amathegi Omkhiqizo

Ukusetshenziswa kanye Nomphumela

I-Pivastatin iyisidakamizwa esilwa ne-hyperlipidemic. Akuyona nje kuphela umuthi omusha, osebenzayo, ophephile, futhi owenziwe ngamakhemikhali okwehlisa ama-lipid osuselwa ku-statin onezindleko eziphezulu kakhulu, kodwa futhi ungumvimbeli onamandla we-3-hydroxy-3-methylglutaryl CoA (HMG-CoA reductase) reductase. Ayigcini nje ngokuba nomthelela omkhulu ekunciphiseni i-LDL-C kanye ne-TC, kodwa futhi ine-polymorphism ebalulekile yezakhi zofuzo, i-bioavailability ephezulu, kanye nengxenye yokuphila isikhathi eside. Futhi bambalwa kuphela abadlula ku-metabolism ye-CYP2C9. Isetshenziselwa ukwelapha i-hyperlipidemia eyinhloko, i-hypercholesterolemia yomndeni, kanye nezinkinga ze-lipid ezixubile.

Isampula Yomkhiqizo

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Ukupakisha Umkhiqizo:

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Ulwazi Olwengeziwe:

Ukwakheka C25H24FNO4
Ukuhlolwa 99%
Ukubukeka Impuphu emhlophe kuya kwengamhlophe
Inombolo ye-CAS 147511-69-1
Ukupakisha 25KG
Impilo Yeshelufu iminyaka engu-2
Isitoreji Gcina endaweni epholile neyomile
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