Ibhande Nomgwaqo: Ukubambisana, Ukuzwana kanye Nokunqoba Nokunqoba
imikhiqizo

Imikhiqizo

Umhlinzeki Womkhiqizi we-Linagliptin CAS: 668270-12-0

I-Linagliptin (amagama okuhweba i-Tradjenta ne-Trajetna) iyisithiyo se-dipeptidyl peptidase-4 (DPP-4) esavunywa yi-US FDA ngoMeyi 2011 ekwelapheni isifo sikashukela sohlobo 2 kanye nokudla nokuzivocavoca. I-Linagliptin (BI-1356) ichazwe njengesithiyo esinamandla kakhulu, esikhetha kancane futhi esisebenza isikhathi eside se-DPP-4. I-Linagliptin yavela emizamweni yokwenza ngcono izithiyo ze-DPP-4 ezisekelwe ku-xanthine kanye nomphumela wokuqala otholakale emkhankasweni we-HTS.


Imininingwane Yomkhiqizo

Amathegi Omkhiqizo

Ukusetshenziswa kanye Nomphumela

I-Linagliptin (TrajentaR, TradjentaTM, TrazentaTM, TrayentaTM) iyisivimbeli somlomo esikhetha kakhulu i-dipeptidyl peptidase-4 futhi iyisidakamizwa sokuqala sekilasi layo esisuswa kakhulu ngendlela engeyona eyezinso. I-Linagliptin iboniswa ukusetshenziswa kanye ngosuku ekwelapheni abantu abadala abanesifo sikashukela sohlobo 2. I-Linagliptin isebenza ukwehlisa amazinga kashukela egazini ngokuvimbela i-enzyme DPP-4, ngaleyo ndlela ivimbele ukuwohloka kwama-hormone e-incretin (i-glucagon-like peptide-1 [GLP-1] kanye ne-glucose-dependent insulinotropic peptide) kanye nokunciphisa ukuphuma kweglucose ngemuva kokudla.

Isampula Yomkhiqizo

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Ukupakisha Umkhiqizo:

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Ulwazi Olwengeziwe:

Ukwakheka C25H28N8O2
Ukuhlolwa 99%
Ukubukeka Impuphu emhlophe
Inombolo ye-CAS 668270-12-0
Ukupakisha 25KG
Impilo Yeshelufu iminyaka engu-2
Isitoreji Gcina endaweni epholile neyomile
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