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Ibandronate Sodium CAS:138844-81-2 Umhlinzeki Womkhiqizi

II-bandronate sodium (i-BONIVA) iyi-bisphosphonate equkethe i-nitrogen evimbela ukumuncwa kwamathambo okubangelwa yi-osteoclast. I-BONIVA iqukethe futhi izithako ezilandelayo ezingasebenzi: i-lactose monohydrate, i-povidone, i-microcrystalline cellulose, i-crospovidone, i-stearic acid ehlanziwe, i-colloidal silicon dioxide, kanye namanzi ahlanziwe. I-tablet film coating iqukethe i-hypromellose, i-titanium dioxide, i-talc, i-polyethylene glycol 6000, kanye namanzi ahlanziwe.


Imininingwane Yomkhiqizo

Amathegi Omkhiqizo

Ukusetshenziswa kanye Nomphumela

I-ibandronate sodium isetshenziswe ukutadisha umphumela wayo ekwandeni nasekuhlelekeni okukhulu kweLeishmania neGiardia ngokukhiqiza ama-concentration curves. Isetshenziswe futhi ukucacisa indlela ama-bisphosphonates aqukethe i-nitrogen (N-BPs) angena ngayo ku-cytosol futhi avimbele umgomo wawo wama-molecule. I-ibandronate sodium ivimbela i-farnesyl diphosphate synthase (IC50 = 20 nM). I-ibandronate sodium nayo iyisithiyo sokuphinda kufakwe amathambo. Ihlolisiswe ngemiphumela yokulwa nomdlavuza ngaphakathi kwe-vitro, njengokungeniswa kwe-apoptosis, ukuvimbela ukukhula kwamaseli, ukuvimbela ukuziphatha okuhlaselayo, kanye nokuvimbela i-angiogenesis kanye nendima yayo ngaphakathi kwe-vivo kumdlavuza ohlukahlukene okuhlanganisa umdlavuza webele nowe-prostate.

Isampula Yomkhiqizo

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Ukupakisha Umkhiqizo:

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Ulwazi Olwengeziwe:

Ukwakheka I-C9H24NNaO7P2
Ukuhlolwa 99%
Ukubukeka Impuphu emhlophe
Inombolo ye-CAS 138844-81-2
Ukupakisha 25KG
Impilo Yeshelufu iminyaka engu-2
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