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I-Somatostatin CAS:51110-01-1
I-Somatostatin iyi-hormone eyenzeka ngokwemvelo evimbela ukukhishwa kwamanye ama-hormone ahlukahlukene emzimbeni. Idlala indima ebalulekile ekulawuleni uhlelo lwe-endocrine futhi ihilelekile ekulawuleni i-hormone yokukhula, i-insulin, i-glucagon, namanye ama-hormone okugaya ukudla.
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I-Linaclotide CAS: 851199-59-2
I-Linaclotide iyi-agonist ye-guanylate cyclase-C ekhonjisiwe ekwelapheni ukuqunjelwa okungapheli kanye ne-irritable bowel syndrome kanye nokuqunjelwa kubantu abadala. Isebenza endaweni yakini endleleni yokugaya ukudla ukwandisa ukukhishwa koketshezi nokusheshisa ukuhamba kwamathumbu, ukunciphisa izimpawu ezihambisana nalezi zimo.
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I-Levosimendan CAS:141505-33-1
I-Levosimendan iyisivuseleli se-calcium kanye nesivuli semisele ye-potassium esisetshenziselwa ukuphatha ukwehluleka kwenhliziyo okubangelwa yi-acute decompensated. Lo muthi unemiphumela ye-inotropic kanye ne-vasodilating, uthuthukisa ukusebenza kwenhliziyo futhi unciphise izimpawu zokwehluleka kwenhliziyo.
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I-Liraglutide CAS:204656-20-2
I-Liraglutide umuthi osetshenziselwa ukwelapha isifo sikashukela sohlobo lwesibili kanye nokukhuluphala. Ingesigaba semithi eyaziwa ngokuthi ama-glucagon-like peptide-1 (GLP-1) receptor agonists, asebenza ngokwandisa ukukhiqizwa kwe-insulin kanye nokunciphisa inani likashukela elikhiqizwa yisibindi. I-Liraglutide itholakala ngendlela yokujova futhi ivame ukunikezwa kanye ngosuku. Umuthi uboniswe ukuthi uyasiza ukwehlisa amazinga kashukela egazini futhi ukhuthaze ukwehla kwesisindo kubantu abanesifo sikashukela sohlobo lwesibili kanye nokukhuluphala.
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I-Octreotide Acetate CAS: 83150-76-9
I-Octreotide acetate iyi-analog ye-octapeptide yokwenziwa ye-hormone yemvelo i-somatostatin. Isebenza njengesivimbeli esinamandla sama-hormone ahlukahlukene nama-neuropeptide, futhi isetshenziswa ekuphatheni izimo ezifana ne-acromegaly, i-carcinoid syndrome, kanye nezinhlobo ezithile zezimila.
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I-Semaglutide CAS:910463-68-2
I-Semaglutide iyi-peptide-1 (GLP-1) receptor agonist efana ne-glucagon esetshenziselwa ukuphathwa kwesifo sikashukela sohlobo 2 kanye nokukhuluphala. Isebenza ngokulawula amazinga kashukela egazini, ukukhuthaza ukwehla kwesisindo, kanye nokunciphisa ingozi yenhliziyo nemithambo yegazi.
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I-Icatibant Acetate CAS:138614-30-9
I-Icatibant acetate umuthi osetshenziselwa ukwelapha i-angioedema yefa (HAE), isimo esingavamile sofuzo esibonakala ngokuvuvukala okungazelelwe nokukhulu kwesikhumba, ulwelwesi lwamafinyila, kanye nezinye izicubu zomzimba. Ingumphikisi we-bradykinin B2 receptor okhethiwe osebenza ngokuvimbela imiphumela ye-bradykinin, umlamuleli oyinhloko wokuvuvukala okuhlobene ne-HAE. I-Icatibant acetate inikezwa ngomjovo ongaphansi kwesikhumba futhi yenzelwe ukuqeda ngokushesha izimpawu zokuhlaselwa yi-HAE okubukhali.
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I-Ganirelix Acetate CAS: 123246-29-7
I-Ganirelix acetate umuthi osetshenziswa kubuchwepheshe bokuzala obusizayo ukuvimbela ukuvuthwa kweqanda ngaphambi kwesikhathi kwabesifazane ababhekene nokucindezeleka okukhulu kwe-ovarian. Ngokucindezela ukukhishwa kwe-hormone ye-luteinizing, i-ganirelix acetate isiza ekuvimbeleni ukukhishwa kweqanda ngaphambi kwesikhathi futhi isekela isikhathi esifanele sokubuyiselwa kwamaqanda ngesikhathi sezinqubo zokukhulelwa kwe-in vitro (IVF). Inikezwa ngemijovo engaphansi kwesikhumba futhi idlala indima ebalulekile ekuphathweni okuphumelelayo kokwelashwa kokungabi nabantwana.
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I-Linaclotide CAS: 851199-59-2
I-Linaclotide iyi-ejenti yokwelapha esetshenziselwa ukwelapha i-irritable bowel syndrome ene-constipation (IBS-C) kanye ne-chronic idiopathic constipation. Njenge-agonist ye-guanylate cyclase-C, i-linaclotide isebenza endaweni yakini emgudwini wokugaya ukudla ukwandisa ukukhishwa koketshezi nokusheshisa ukuhamba kwamathumbu, ngaleyo ndlela inciphise izimpawu ezifana ne-constipation kanye nokungakhululeki kwesisu.
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I-Ziconotide Acetate CAS:107452-89-1
I-Ziconotide acetate iyinguqulo yokwenziwa ye-peptide compound ethathwe ebuchosheni be-Conus magus snail. Isetshenziswa njengomuthi wokudambisa ubuhlungu wokuphatha ubuhlungu obukhulu obungapheli ezigulini ezingabekezeleli noma ezingaphendulanga kwezinye izindlela zokwelapha. I-Ziconotide acetate inikezwa ngokufaka ngaphakathi kwe-thecal, okuhlinzeka impumuzo eqondiwe kubantu ababhekene nezimo zobuhlungu obungalawuleki.
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I-Degarelix CAS:214766-78-6
I-Degarelix iyi-gonadotropin-releasing hormone (GnRH) receptor antagonist esetshenziswa ekwelapheni umdlavuza we-prostate othuthukile. Isebenza ngokucindezela ngokushesha ukukhiqizwa kwe-testosterone, i-hormone ekhuthaza ukukhula kwezimila ze-prostate.
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I-Acetyl Octapeptide-3/1 CAS:868844-74-0
I-Acetyl Octapeptide-3, eyaziwa nangokuthi i-Argireline, iyi-peptide yokwenziwa evame ukusetshenziswa emikhiqizweni yokunakekelwa kwesikhumba ngenxa yezakhiwo zayo zokulwa nokuguga. Le peptide kukholakala ukuthi isebenza ngokunciphisa ukufinyela kwemisipha, okungasiza ekunciphiseni ukubonakala kwemigqa emincane nemibimbi, ikakhulukazi ezindaweni ezivame ukuba nemigqa yokubonakaliswa njengebunzi kanye naseduze kwamehlo.
