Ibhande Nomgwaqo: Ukubambisana, Ukuzwana kanye Nokunqoba Nokunqoba
imikhiqizo

Imikhiqizo

I-Delamanid CAS:681492-22-8

I-Delamanid umuthi we-antimycobacterial ohlukaniswe njenge-diarylquinoline derivative, osetshenziswa kakhulu ekwelapheni isifo sofuba esingamelana nemithi eminingi (i-MDR-TB). Isebenza ngokugxila ku-mycobacterial ATP synthase, okuholela ekuphazamisekeni kokukhiqizwa kwamandla kumagciwane abangela isifo sofuba. I-Delamanid ibhekwa njenge-ejenti yomugqa wesibili yamacala e-MDR-TB lapho kukhona ukumelana nemithi yomugqa wokuqala evamile. Lo muthi utholakala ngesimo sethebhulethi futhi uvame ukunikezwa njengengxenye yohlelo oluphelele lokulwa nokutheleleka kwesifo sofuba okungamelana nemithi.


Imininingwane Yomkhiqizo

Amathegi Omkhiqizo

Ukusetshenziswa kanye Nomphumela:

I-Delamanid iyithuluzi elibalulekile lezokwelapha ekuphathweni kwesifo sofuba esingamelana nemithi eminingi, uhlobo olubi lwesifo sofuba olungaphenduli ekwelashweni okujwayelekile komugqa wokuqala. Ngokuvamile ifakwa ezinhlotsheni zokwelapha ezihlanganisiwe ze-MDR-TB ukuze kuthuthukiswe imiphumela yokwelashwa futhi kuncishiswe ingozi yokuthuthukiswa kokumelana nemithi. Abahlinzeki bezempilo banikeza i-delamanid kanye neminye imithi yokulwa nesifo sofuba yomugqa wesibili ngokusekelwe ezicini zesiguli ngasinye, okuhlanganisa ubukhulu bokumelana nemithi, umlando wokwelashwa wangaphambilini, kanye nesimo sempilo iyonke. Umuthi uvame ukunikezwa ngomlomo ngesimo sethebhulethi, kanye nokuvama komthamo kanye nobude besikhathi obuhambisana nezidingo ezithile zesiguli ngasinye. Iziguli ezelashwa nge-delamanid ziyalulekwa ukuthi zinamathele ngokuqinile ohlelweni olubekiwe, njengoba ukudla njalo imithi kubalulekile ekufezeni impumelelo yokwelapha kanye nokunciphisa ingozi yokwehluleka kokwelashwa. Ukuqapha njalo imiphumela emibi engaba khona, njengokuphazamiseka kwesisu noma izinguquko ekusebenzeni kwesibindi, kubalulekile ngesikhathi sokwelashwa. Ukwelashwa nge-Delamanid kuvame ukuqaliswa futhi kuqondiswe ochwepheshe bezempilo abanolwazi ekuphatheni amacala ofuba angamelana nemithi. Ukubambisana phakathi kwethimba lezempilo nesiguli kubalulekile ukuqinisekisa ukulandelwa kokwelashwa, ukuqapha inqubekela phambili, kanye nokubhekana nanoma yiziphi izinkinga noma izinkinga ngokushesha. Ekuphetheni, i-delamanid idlala indima ebalulekile ekulweni nesifo sofuba esingamelana nemithi eminingi, inikeza iziguli nabahlinzeki bezempilo inketho yokwelapha ephumelelayo yokulwa nalesi sifo esithathelwanayo esiyinselele nokuvimbela ukusabalala kwaso emiphakathini.

Isampula Yomkhiqizo:

I-L-Arginine1
I-L-Arginine2

Ukupakisha Umkhiqizo:

I-L-Arginin3

Ulwazi Olwengeziwe:

Ukwakheka C25H25F3N4O6
Ukuhlolwa 99%
Ukubukeka impuphu emhlophe
Inombolo ye-CAS 681492-22-8
Ukupakisha Encane futhi enkulu
Impilo Yeshelufu iminyaka engu-2
Isitoreji Gcina endaweni epholile neyomile
Isitifiketi I-ISO.

 


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